Research Paper (721)

  • Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists
    Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists

    Tsotinis A.

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  • Mechanism of thienopyridone and iminothienopyridinedione inhibition of protein phosphatases
    Mechanism of thienopyridone and iminothienopyridinedione inhibition of protein phosphatases

    Zhang Z.

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  • Fluoroquinolone-derived fluorescent probes for studies of bacterial penetration and efflux
    Fluoroquinolone-derived fluorescent probes for studies of bacterial penetration and efflux

    Stone M.R.L.

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  • Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen
    Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen

    Atkinson B.N.

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  • Synthesis, ribosomal selectivity, and antibacterial activity of netilmicin 4?-derivatives
    Synthesis, ribosomal selectivity, and antibacterial activity of netilmicin 4?-derivatives

    Sonousi A.

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  • Synthesis of novel vanillin derivatives: Novel multi-targeted scaffold ligands against Alzheimer's disease
    Synthesis of novel vanillin derivatives: Novel multi-targeted scaffold ligands against Alzheimer's disease

    Scipioni M.

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  • 3D QSAR-based design and liquid phase combinatorial synthesis of 1,2-disubstituted benzimidazole-5-carboxylic acid and 3-substituted-5 H-benzimidazo[1,2-d] [1,4]benzodiazepin-6(7 H)-one derivatives as anti-mycobacterial agents
    3D QSAR-based design and liquid phase combinatorial synthesis of 1,2-disubstituted benzimidazole-5-carboxylic acid and 3-substituted-5 H-benzimidazo[1,2-d] [1,4]benzodiazepin-6(7 H)-one derivatives as anti-mycobacterial agents

    Sitwala N.D.

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  • Affinity of fentanyl and its derivatives for the ?1-receptor
    Affinity of fentanyl and its derivatives for the ?1-receptor

    Lipi?ski P.F.J.

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  • Synthesis of DNA-coupled isoquinolones and pyrrolidines by solid phase ytterbium- A nd silver-mediated imine chemistry
    Synthesis of DNA-coupled isoquinolones and pyrrolidines by solid phase ytterbium- A nd silver-mediated imine chemistry

    Potowski M.

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  • Gramicidin S-inspired antimicrobial cyclodextrin to disrupt gram-negative and gram-positive bacterial membranes
    Gramicidin S-inspired antimicrobial cyclodextrin to disrupt gram-negative and gram-positive bacterial membranes

    Yamamura H.

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  • The winding road of the uvaretin class of natural products: From total synthesis to bioactive agent discovery
    The winding road of the uvaretin class of natural products: From total synthesis to bioactive agent discovery

    Dallman J.

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  • Derivatisation of parthenolide to address chemoresistant chronic lymphocytic leukaemia
    Derivatisation of parthenolide to address chemoresistant chronic lymphocytic leukaemia

    Li X.

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  • Synthesis of endolides A and B: Naturally occurring N-methylated cyclic tetrapeptides
    Synthesis of endolides A and B: Naturally occurring N-methylated cyclic tetrapeptides

    Davison E.K.

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  • Piperidine carbamate peptidomimetic inhibitors of the serine proteases HGFA, matriptase and hepsin
    Piperidine carbamate peptidomimetic inhibitors of the serine proteases HGFA, matriptase and hepsin

    Damalanka V.C.

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  • Binding site characterization-similarity, promiscuity, and druggability
    Binding site characterization-similarity, promiscuity, and druggability

    Ehrt C.

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  • Novel carbohydrate modified berberine derivatives: Synthesis and: In vitro anti-diabetic investigation
    Novel carbohydrate modified berberine derivatives: Synthesis and: In vitro anti-diabetic investigation

    Han L.

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  • Synthesis of bicyclic 1,4-thiazepines as novel anti-: Trypanosoma brucei brucei agents
    Synthesis of bicyclic 1,4-thiazepines as novel anti-: Trypanosoma brucei brucei agents

    Vairoletti F.

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  • A MedChem toolbox for cereblon-directed PROTACs
    A MedChem toolbox for cereblon-directed PROTACs

    Steinebach C.

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  • Non-lethal growth inhibition by arresting the starch utilization system of clinically relevant human isolates of: Bacteroides dorei
    Non-lethal growth inhibition by arresting the starch utilization system of clinically relevant human isolates of: Bacteroides dorei

    Santilli A.D.

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  • Druggability assessment of mammalian Per-Arnt-Sim [PAS] domains using computational approaches
    Druggability assessment of mammalian Per-Arnt-Sim [PAS] domains using computational approaches

    De Souza J.V.

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  • A cell-based screening system for RNA polymerase i inhibitors
    A cell-based screening system for RNA polymerase i inhibitors

    Tan X.

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  • Biochemical and microbiological evaluation of: N-aryl urea derivatives against mycobacteria and mycobacterial hydrolases
    Biochemical and microbiological evaluation of: N-aryl urea derivatives against mycobacteria and mycobacterial hydrolases

    Vartak A.

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  • The synthesis and biological evaluation of novel gardenamide A derivatives as multifunctional neuroprotective agents
    The synthesis and biological evaluation of novel gardenamide A derivatives as multifunctional neuroprotective agents

    Zhang Z.

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  • Design, synthesis and biological evaluation of ?-peptoid-capped HDAC inhibitors with anti-neuroblastoma and anti-glioblastoma activity
    Design, synthesis and biological evaluation of ?-peptoid-capped HDAC inhibitors with anti-neuroblastoma and anti-glioblastoma activity

    Re?ing N.

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  • New methods to assess 6-thiopurine toxicity and expanding its therapeutic application to pancreatic cancer via small molecule potentiators
    New methods to assess 6-thiopurine toxicity and expanding its therapeutic application to pancreatic cancer via small molecule potentiators

    Weeramange C.

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  • Synthesis and direct comparison of the anticancer activities of phomopsolides D and e and two 7-oxa-/7-aza-analogues
    Synthesis and direct comparison of the anticancer activities of phomopsolides D and e and two 7-oxa-/7-aza-analogues

    Aljahdali A.Z.

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  • Evaluation of anti-inflammatory activity and molecular docking study of new aza-bicyclic isoxazoline acylhydrazone derivatives
    Evaluation of anti-inflammatory activity and molecular docking study of new aza-bicyclic isoxazoline acylhydrazone derivatives

    Mota F.V.B.

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  • Methyl sulfonamide substituents improve the pharmacokinetic properties of bicyclic 2-pyridone based: Chlamydia trachomatis inhibitors
    Methyl sulfonamide substituents improve the pharmacokinetic properties of bicyclic 2-pyridone based: Chlamydia trachomatis inhibitors

    Kulen M.

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  • Development of hydroxamate-based histone deacetylase inhibitors of bis-substituted aromatic amides with antitumor activities
    Development of hydroxamate-based histone deacetylase inhibitors of bis-substituted aromatic amides with antitumor activities

    Ge D.

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  • Synthesis and biological evaluation of structurally diverse ?-conformationally restricted chalcones and related analogues
    Synthesis and biological evaluation of structurally diverse ?-conformationally restricted chalcones and related analogues

    Maguire C.J.

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